中文名称: | 盐酸利多卡因 促销 | ||||
---|---|---|---|---|---|
英文名称: | Lidocaine Hydrochloride | ||||
别名: | 盐酸利多卡因一水合物 LidocaLidocaine Hydrochlorideine hydrochloride monohydrate | ||||
CAS No: | 6108-05-0 | 分子式: | C14H22N2O.HCl.H2O | 分子量: | 288.81 |
CAS No: | 6108-05-0 | ||||
分子式: | C14H22N2O.HCl.H2O | ||||
分子量: | 288.81 | ||||
MDL: | MFCD00150329 |
包装规格:
5mg 10mg 25mg 50mg 100mg in glass bottle
产品简介:
Lidocaine (Lignocaine) hydrochloride hydrate 抑制涉及复杂电压和依赖性的钠通道 (sodium channels)。Lidocaine hydrochloride hydrate 通过调节 miR-145 表达和进一步抑制 MEK/ERK 和 NF-κB 信号通路来减少胃癌细胞的生长,迁移和侵袭。Lidocaine hydrochloride hydrate 是一种酰胺衍生物,可用于研究室性心律失常。
靶点:
ERK
NF-κB
MEK
NF-κB
MEK
体外研究:
Lidocaine (Lignocaine) (10 nM; 48 hours) decreases significantly cell proliferation.
Lidocaine (1-10 nM; 24-72 hours) inhibits cell viability and achieves the most suppressing effects at the concentration of 10 nM and treatment time 48 hours.
Lidocaine (10 nM; 48 hours) increases significantly the apoptotic cell rate.
Lidocaine (10 nM; 48 hours) down-regulates Cyclin D1 and up-regulates p21 expression significantly.
Lidocaine (1-10 nM; 24-72 hours) inhibits cell viability and achieves the most suppressing effects at the concentration of 10 nM and treatment time 48 hours.
Lidocaine (10 nM; 48 hours) increases significantly the apoptotic cell rate.
Lidocaine (10 nM; 48 hours) down-regulates Cyclin D1 and up-regulates p21 expression significantly.
体内研究:
Lidocaine (Lignocaine) causes completely reversible tail nerve block in rats. Mechanical nociception block produced by lidocaine has slower onset and faster recovery compared with thermal nociception block.
保存条件:
-20°C
注意事项:
1、为了您的安全和健康,请穿实验服并戴一次性手套操作。
2、以上信息仅做参考交流之用。
2、以上信息仅做参考交流之用。
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参考文献 & 客户发表文献
本计算器可帮助您计算出特定溶液中溶质的质量、溶液浓度和体积之间的关系,公式为:
质量 (g) = 浓度 (mol/L) x 体积 (L) x 分子量 (g/mol)
摩尔浓度计算公式
用本工具协助配置特定浓度的溶液,使用的计算公式为:
开始浓度 x 开始体积 = 最终浓度 x 最终体积
稀释公式
稀释公式一般简略地表示为:C1V1 = C2V2 ( 输入 输出 )