参考文献
1: Adams ML, Sharma V, Gokhale M, Huang Y, Stefanski K, Su C, Hussain MA.
Dehydration and Stabilization of a Reactive Tertiary Hydroxyl Group in Solid Oral
Dosage Forms of BMS-779788. J Pharm Sci. 2016 Apr;105(4):1478-88. doi:
10.1016/j.xphs.2015.12.028. Epub 2016 Feb 23. PubMed PMID: 26921118.
2: Kirchgessner TG, Martin R, Sleph P, Grimm D, Liu X, Lupisella J, Smalley J,
Narayanan R, Xie Y, Ostrowski J, Cantor GH, Mohan R, Kick E. Pharmacological
characterization of a novel liver X receptor agonist with partial LXRα activity
and a favorable window in nonhuman primates. J Pharmacol Exp Ther. 2015
Feb;352(2):305-14. doi: 10.1124/jpet.114.219923. Epub 2014 Dec 2. PubMed PMID:
25467132.
3: Kick E, Martin R, Xie Y, Flatt B, Schweiger E, Wang TL, Busch B, Nyman M, Gu
XH, Yan G, Wagner B, Nanao M, Nguyen L, Stout T, Plonowski A, Schulman I,
Ostrowski J, Kirchgessner T, Wexler R, Mohan R. Liver X receptor (LXR) partial
agonists: biaryl pyrazoles and imidazoles displaying a preference for LXRβ.
Bioorg Med Chem Lett. 2015 Jan 15;25(2):372-7. doi: 10.1016/j.bmcl.2014.11.029.
Epub 2014 Nov 15. PubMed PMID: 25435151.