2020-10-20
1: Barsyte-Lovejoy D, Li F, Oudhoff MJ, Tatlock JH, Dong A, Zeng H, Wu H, Freeman 
SA, Schapira M, Senisterra GA, Kuznetsova E, Marcellus R, Allali-Hassani A, 
Kennedy S, Lambert JP, Couzens AL, Aman A, Gingras AC, Al-Awar R, Fish PV, 
Gerstenberger BS, Roberts L, Benn CL, Grimley RL, Braam MJ, Rossi FM, Sudol M, 
Brown PJ, Bunnage ME, Owen DR, Zaph C, Vedadi M, Arrowsmith CH. (R)-PFI-2 is a 
potent and selective inhibitor of SETD7 methyltransferase activity in cells. Proc 
Natl Acad Sci U S A. 2014 Sep 2;111(35):12853-8. doi: 10.1073/pnas.1407358111. 
Epub 2014 Aug 18. PubMed PMID: 25136132; PubMed Central PMCID: PMC4156762.